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Nitrogen Rich Heterocycles - Coggle Diagram
Nitrogen Rich
Heterocycles
1. Design and Synthesis
Benzamides
Tetrazoles
N-Acyl carbothioamides
Triazolone hybrids
Chalcones
Triazolothione hybrids
Sulphonamides
Thiazolyl-2-hdrazines
Hydrazide-Schiff Bses
Thieno[2,3-b]pyridine-2-carboxamides
2. Work Up
Recrystallization
Column Chromatography
Appearance (Color)
Filteration
Melting Points
Miscibility
Rf Values
3. Characterization
NMR
Mass
FT-IR
X-ray Diffraction
CHNS Analysis
4. In Silico Analysis
Structure Activity Relationships
Drug-Likeness
Dynamic Simulations
Hirschfeld Surface Analysis
Molecular Docking
GOLD Analysis
CHEMPLP
CHEMSCORE
GOLDCORE
ASP CORE
DFT Calculation
5. In Vitro Evaluation
Antimicrobial Assay
Antifungal Assay
Antileishmanial Assay
Antibacterial Assay
DNA Cleavage Assay
Antidiabetic Assay
Alpha-Glucosidae
Alpha-Amylase
AntiCancer Assay
Alkaline Phosphatase Assay
h-IAP
h-TNAP
Anti-Oxidant Assay
DPPH
Nitric Oxide
Hydroxyl
Iron Chelation
TAC/TRP