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Nitrogen Rich Heterocycles : - Coggle Diagram
Nitrogen Rich Heterocycles
:
1. Design and Synthesis
N-Acyl carbothioamides
Benzamides
Triazolone hybrids
Tetrazoles
Triazolothione hybrids
Chalcones
Thiazolyl-2-hdrazines
Sulphonamides
Thieno[2,3-b]pyridine-2-carboxamides
Hydrazide-Schiff Bses
2. Work Up
Appearance (Color)
Recrystallization
Melting Points
Column Chromatography
Rf Values
Filteration
Miscibility
4. In Silico
Analysis
Molecular Docking
Dynamic Simulations
Structure Activity Relationships
Drug-Likeness
GOLD Analysis
GOLD Score
ASP Score
CHEMPLP
CHESCORE
Hirshfeld Surface Analysis
5. In Vitro
Assay
DNA Ladder
Anticancer
Alpha-Amylase
Alkaline Phosphatase Inhibition
Alpha-Glucosidase
hRBCs Hemolysis
Anti-oxidant
Iron Chelating
DPPH Scavenging
Nitric Oxide
Hydroxyl Scavenging
TAC/TRP
Brine Shrimp Lethality
Antimicrobial
Antifungal
**Antileishmanial
Antibacterial
3. Characterization
CHNS Analysis
NMR Spectroscopy
Mass Spectrometry
FT-IR Spectroscopy
X-ray Diffraction