Please enable JavaScript.
Coggle requires JavaScript to display documents.
SEROTONIN AND RELATED DRUGS, C/I:- with Ergotamine, S/E:- Coronary…
SEROTONIN AND RELATED DRUGS
5HT1 Agonists
5HT 1B/1D Agonist
Triptans
Frava
triptan
Nara
triptan
Riza
triptan
Suma
triptan
Zolmi
triptan
Ele
triptan
Almo
triptan
5HT1F Agonists
Acts on Gi
Decrease CGRP release in 5th Cranial nerve
Prevent meningeal vessel dilation
used in Acute Attack of Miagraine
5HT1A Agonist
Decrease 5HT release
Anxiolytic
Buspirone (Used in smoking cessation)
Ipsapirone
Gepirone
5HT4 Agonist
Mosapride
Cisapride
Metoclopramide
Increase Peristalisis
Prokinetic drug
Used in Gastroesophageai Reflex Disease (GERD)
5HT3 Agonist
Ondan
setron
Palano
setron
Dolo
setron
Topo
setron
Grani
setron
MOA
Block CTZ Area
Antiemetic
DOC for Chemotherapy induced Nausea and Vomiting
5HT2
Agonist
Locaserin (for obesity)
now banned
Due to risk of Cancer
LSD
Antagonist
Cyproheptadine
Methysergide
Pizotifen
Fibanserin
(
Uses :-
Migraine Prophylaxis,
Serotonin Syndrome)
Atypical Antipsychotics
Clozapine
Olanzapine
Quetiapine
C/I:
- with Ergotamine
Potent Vasocontrictor
Gangrene of Organ with endarteries
S/E:
-
Coronary Vasoconstriction
Sweating
Pain in Jaw/ Neck
(Gs)
(Gi)
(
Gq
)
Ligand-Gated ion channel [Na+/Ca2+]