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drug for GI, Laxative瀉藥, 蠕動促進劑, 止吐藥物, 止瀉藥, 腸躁症(IBS)用藥 - Coggle Diagram
drug for GI
antibiotic
抑制胃幽門桿菌
Amoxicillin
Clarithromycin
Metronidazole
少用
牙科常用藥
Tetracyline
antacids
NaHCO3
Mg(OH)2
腹瀉
Al(OH)3
便秘
CaCO3
Anticholinergics(M)
non-selective
-pine
Atropine
specific
-zepine
Pirenzepine
Telenzepine
block M1 receptor
block ECL cell
Proton pump inhibitor (PPI)
阻斷H-K ATPase
抑制胃酸效果最佳
-prazole
Omeprazole
Esomeprazole
Lansoprazole
Rabeprazole
Pantoprazole
treat
消化性潰瘍
出血消化性潰瘍
胃食道逆流
mucosa protect agent
Sucralfate
Colloidal bismuth compounds
能抑制H. pylori生長
H2 receptor blocker
-tidine
Cimetidine
交互作用最多
抑制CYP
Ranitidine
Famotidine
Nizatidine
treat
消化性潰瘍
被PPI取代
胃食道逆流
Postaglandin analogs
Misoprostol
PGE1 類似物
抑制酸分泌
刺激子宮收縮
和RU-486並用
墮胎
胃酸抑制劑
Laxative瀉藥
滲透性瀉劑
Sorbitol
Lactulose
treat急性門系肝腦病變
Polyethylene Glycol(PEG)
刺激&興奮劑
Castol oil蓖麻油
造成宮縮
含ricinoleic acid
Bisacody
治療便秘最常使用
Opioid receptor antagonists
Methylnaltrexone
Alvimopan
膨脹性瀉劑
Psyllium車前子
天然製劑
氯離子通道活化劑
Lubiprostone
PGE1類似物
蠕動促進劑
Dopamine(D2) receptor antagonist
Metoclopramide
能過BBB
cause 錐體外症狀(帕金森氏症)
增加血清泌乳素
漏奶症
男性女乳症
Doperidone
不會過BBB
抑制膽鹼性平滑肌刺激
強制胃排空
抗噁心、止吐
Motilin receptor agonist
Motilin
Macrolides antibotics
Erythromycin
Azithromcyin
Cholinomimetic agent
Bethanechol
Neostigmine
Serotonin antagonist/agonist
-pride
Cisapride
5-HT4 agonist
心律不整
CYP3A4 substrate
不能和ketoconazole、erythromycin並用
Mosapride
selective 5-HT4 agonist
treat糖尿病胃輕癱
止吐藥物
H1 Antihistamines & Anticholinergic Drug
預防、治療動暈症
H1 Antihistamines
Diphenhydramine、Dimenhydrinate
Meclizine
較少鎮靜作用
Anticholinergic
Hyoscine/Scopolamine
最有效藥物
5-HT3 receptor antagonist
-setron
Ondansetron
Granisetron
Dolasetron
Palonosetron
預防急性化療引起的噁心嘔吐
Neurokinin(NK1) receptor antagonist
-pitant
Aperpitant
Fosaprepitant
Dopamine-receptor antagonist
-azine
Chlorpromazine
臨床有使用
Prochlorperazine
止瀉藥
Opioid agonists
Loperamide
臨床常用止瀉藥物
無CNS影響
不會成癮
Diphenoxylate
else
腸躁症(IBS)用藥
5-HT4 receptor agonist
Tegaserod
治便祕
造成腹瀉
Prucalopride
5-HT3 receptor antagonist
Alosetron
治腹瀉
造成便秘