Wnt Signaling

Pathways

Non canonical pathway

Planar cell polarity

Calcium pathway

Int1(Wnt1)

Canonical pathway

Wingless gene

β-catenin

APC gene

T-cell factor

Cancer

Role in cancer

Melanoma

Breast cancer

Leukemia

Gastrointestinal/Colo-rectal cancer

Metastasis

Treatment and clinical trials

Epithelial to mesenchymal transition

SNAI2

Induce formation

Fdz2

ASPP2

PI3K-Akt signaling

Cause tumor cells to metastasise

High levels β-catenin

Loss of APC

Over expression of WNT ligands

Wnt canonical pathway delaying senescence of melanocytes

Regulation of gene transcription

Independent of β-catenin

Dependent on β-catenin

Regulates cytoskeleton

Regulates cytoskeleton

Anti-Wnt secretion

Drugs to target Wnt ligands and receptors

Immune checkpoint blockade

Anti-CTLA4 and anti-PD-L1

Monoclonal antibodies

LGK974

OMP-54F28

OMP18R5