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Everolimus (Side effects (Diarrhoea, Esophagitis, Fatigue, Stomatitis,…
Everolimus
Side effects
Diarrhoea
Esophagitis
Fatigue
Stomatitis
Stomach cramps
Rash,itchy or dry skin
Contraindications
Kidney problems
High cholesterol
Diabetes
Cancer
Anaemua
Indications
To treat various types of cancer such as lung,kidney,breast cancer etc.
Used in people with tuberous sclerosis complex to treat certain types of benign tumors
Mechanism of action
It binds to its protein receptor FKBP12
This protein directly interacts with mTORC1 and inhibit its downstream signaling
Storage
Stored at room temperature
Route of administration
Oral