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Pituitary Drugs (Ergot-derived Da agonists (Bromocriptine Cabergoline …
Pituitary Drugs
Ergot-derived Da agonists
Bromocriptine
Cabergoline
Pergolide
SE
Fibrosis
GI upset: esp. nausea
Postural hypotension
Drowsiness
Neuropsych syndromes
CI
Cardiovascular disease
Porphyria
Psychosis
Levels ↑d by:
octreotide
macrolides
Use
prolactinoma
acromegaly
Monitor heart with echo
Somatostatin analogues
Octreotide
Lanreotide
SE
Diarrhoea
Gallstones
Use
acromegaly
carcinoid syndrome
GH receptor antagonist
Pegvisomant
Use
acromegaly
11β-hydroxylase inhibitor
inhibits adrenal cortisol
production
Metyrapone
SE
Hypoadrenalism
Use
Cushing’s syndrome particularly if resistant to surgery