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Oral Hypoglycaemics (Gliclazide (s)
Tolbutamide (s)
Glipizide (s)
…
Oral Hypoglycaemics
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Metformin
MOA
Biguanide
Insulin sensitizer
- ↓ gluconeogenesis
- ↑ peripheral glucose use
- ↓ LDL and VLDL
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Pioglitazone
MOA
Thiazolidinedione
Peripheral insulin sensitizer
PPAR gamma ligand (nuclear receptor
involved in glucose and lipid homeostasis)
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-
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Acarbose
MOA
Intestinal α-glucosidase inhibitor
Delays carb absorption → ↓ post-prandial
blood glucose
Little effect on fasting glucose
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Exenatide
Liraglutide
MOA
Insulin secretagogue
GLP-1 analogue
- ↑ insulin secretion and sensitisation
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