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indirect (Blocker (抑制合成、儲存、釋放) (Hemicholinium (抑制神經攝入choline), Botulism…
indirect
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Stimulator (抑制AChE)
Nicotinic Receptor
Edrophonium (short, 診斷MG)
Both
Neostigmine (腸麻痺、尿滯留、Tubocurarine 過量、MG), Physostigmine (青光眼、BBB、Atropine過量、MG)
direct
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Antagonist
Muscarinic (四級周邊、三級中樞)
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眼科
Atropine(長效), Tropicamide(短效), Homatropine
腸胃科
Pirezapine(不便秘), Propenthiline(四級胺、便秘)(皆抑胃酸分泌 M1 R)
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-
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Nicotinic (為鬆弛肌肉)
中樞型
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Baclofen(GABAb,open K channel)
其他
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Tubocurarine, Pancuronium (競爭ACh R、Neostigmine解毒)
Succinylcholine, Decamethonium (去極化、IF惡性體溫升高-> Dantrolene)