indirect

direct

Blocker (抑制合成、儲存、釋放)

Stimulator (抑制AChE)

Nicotinic Receptor

Both

Hemicholinium (抑制神經攝入choline)

Botulism (抑制小泡釋放)

Edrophonium (short, 診斷MG)

Neostigmine (腸麻痺、尿滯留、Tubocurarine 過量、MG), Physostigmine (青光眼、BBB、Atropine過量、MG)

Antagonist

Agonist

Muscarinic (四級周邊、三級中樞)

Nicotinic (為鬆弛肌肉)

Muscarinic

Nicotinic

耳鼻喉

胸內

眼科

腸胃科

神內

泌尿

中樞型

其他

Pilocarpine(縮瞳-青光眼)

Methacholine (診斷氣喘)

Bethanecol (腸麻痺、尿滯留)

Succinylcholine (先收縮再癱瘓肌肉)

Diazepam (GABAa)

Baclofen(GABAb,open K channel)

Dantrolene (抑鈣從肌漿網出)

Tubocurarine, Pancuronium (競爭ACh RNeostigmine解毒)

Succinylcholine, Decamethonium去極化IF惡性體溫升高-> Dantrolene

Benztropine (Parkinson's)

Atropine(長效), Tropicamide(短效), Homatropine

Scopolamine(暈車藥)

Ipatropium (四級胺、for COPD [with B blocker]、吸入)

Pirezapine(不便秘), Propenthiline(四級胺、便秘)(皆抑胃酸分泌 M1 R)

Clidinium (腸躁症)

Oxybutinin (尿失禁)

Both

Nicotine

Carbachol (縮瞳-青光眼)

ACh