indirect
direct
Blocker (抑制合成、儲存、釋放)
Stimulator (抑制AChE)
Nicotinic Receptor
Both
Hemicholinium (抑制神經攝入choline)
Botulism (抑制小泡釋放)
Edrophonium (short, 診斷MG)
Neostigmine (腸麻痺、尿滯留、Tubocurarine 過量、MG), Physostigmine (青光眼、BBB、Atropine過量、MG)
Antagonist
Agonist
Muscarinic (四級周邊、三級中樞)
Nicotinic (為鬆弛肌肉)
Muscarinic
Nicotinic
耳鼻喉
胸內
眼科
腸胃科
神內
泌尿
中樞型
其他
Pilocarpine(縮瞳-青光眼)
Methacholine (診斷氣喘)
Bethanecol (腸麻痺、尿滯留)
Succinylcholine (先收縮再癱瘓肌肉)
Diazepam (GABAa)
Baclofen(GABAb,open K channel)
Dantrolene (抑鈣從肌漿網出)
Tubocurarine, Pancuronium (競爭ACh R、Neostigmine解毒)
Succinylcholine, Decamethonium (去極化、IF惡性體溫升高-> Dantrolene)
Benztropine (Parkinson's)
Atropine(長效), Tropicamide(短效), Homatropine
Scopolamine(暈車藥)
Ipatropium (四級胺、for COPD [with B blocker]、吸入)
Pirezapine(不便秘), Propenthiline(四級胺、便秘)(皆抑胃酸分泌 M1 R)
Clidinium (腸躁症)
Oxybutinin (尿失禁)
Both
Nicotine
Carbachol (縮瞳-青光眼)
ACh