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CYP-p450 :fire: (CYP3A4 (Substrater (Lipidstofskiftet (Fibrater, Statiner …
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CYP-p450 :fire:
CYP3A4
Induktorer
Fenytoin, karbamazepin, barbiturater, rifampicin, perikum (naturmedicin)
Inhibitorer
Makrolidantibiotika, keto/flukonazol, verapamil - diltiazem, grapefrugt juce, metoklopramid, p-piller, allopurinol
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CYP1A2
Induktorer:
Rifampicin, karbamazepin, fenytoin (3 af de samme som for CYP 3A4)
Inhibitorer
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Virus/bakterier
Makrolider som erythromycin, clarithyromycin
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CYP2C9
Induktorer
3 af de samme som for CYP3A4: karbamazepin, rifampicin, perikum
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