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ANS Pharmacological Classification - Coggle Diagram
ANS Pharmacological Classification
PNS
Cholinergic Drugs
Agonists
Choline esters
Acetylcholine
Methacholine
Bethanechol
Alkaloids
Muscarine
Pilocarpine
Anticholinestearses
Reversible
Carbamates
Physostigmine
Neostigmine
Pyridostigmine
Non-carbamates
Edrophonium
Tacrine
Galantamine
Irreversible
Carbamates
Insecticides : Sevin, Baygon
Organophosphates
Dyflos (DFP)
Echothiophate
Insecticides :Malathion
Nerve Gas
Anti Cholinergic Drugs
Natural/ Non selective
Atropine
Hyoscine = Scopolamine
Selective
M1
Benz-tropine
Benz-hexol = Trihexyphenydyl
M3
Glycopyrolate
Tropicamide
Cyclopentolate
Ipratropium
Tiotropium
Oxybutynin
SNS
Adrenergic Drugs
Indirectly acting
Reuptake inhibitor
Cocaine
Modafinil
Atomoxetine
Sibutramine
Increase NA release
Tyramine
Amphetamine
Directly acting
Non catecholamines
a1 agonist
phenylephrine
xylometazoline or oxymetazoline
a2 agonist
Clonidine
Methyl dopa
b2 agonist
Salbutamol
Salmeterol
Tocolytics= uterine relaxants
b1 agonist
Dobutamine
Catecholamines
DA
Dobutamine
Fenaldopam
Adrenaline
NA
Isopranaline
Mixed
Ephedrine
Anti Adrenergic Drugs
alpha blocker
Non selective
Phenoxybenzamine
Phentolamine
selective = a1 blocker
Prazosin
beta blocker
Non selective /1st gen
Propranolol
Sotalol
Timolol
Pindolol
Cardioselective / 2nd gen/ b1 blocker
Metoprolol
Atenolol
a+b blocker
Labetalol
Carvedilol
for Glaucoma
beta blocker
Timolol
CA i
Acetazolamine(oral/IV)
Brinzolamaine
a2 agonist
Apraclonidine
Miotic
Pilocarpine
For Narrow Angle Glaucoma
DOC: Acteazolamide
I. V. Mannitol
Topical E/D
Receptors in
PNS
Cholinergic transmission
Ion Channel type
N
Nm
NMJ
Nn
CNS Neurons
GPCR
M
Gi / Go
M2
Heart
Gq
M3
Smooth Muscle and Glands
M1
CNS GIT
SNS
Adrenergic transmission
Alpha
Gq
a1
Prostate
BV
Eye
Sphincter GIT
Sphincter Bladder
Gi
a2
Presynaptic neuron in CNS
Beta
b1
Heart
JG cells
b2
Smooth Muscle
Skeletal muscle spindle
Liver
Cell surface for k bal
b3
Adipocytes
Bladder