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藥理 (免疫藥物 (抑制基因而抑制發炎反應:Glucocorticoids (prednisolone→prednisone,…
藥理
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Anti-cancer
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Chemotherapy
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Anti-Metabolites
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pyrimidine:Fluorouracil(5-FU)→在體內會變成FdUMP→與MTHF(one carbon donor)、Thymidylate synthase結合抑制活性
→使dUMP無法變成dTMP
Front-line:5-FU+leucovorin
葉酸類:Methotrexate(MTX)→抑制DHFR→抑制one-carbon donor形成→抑制核苷酸生成
適用:乳癌(CMF)、ALL、Choriocarcinoma
使用Leucovorin可以減緩副作用
Cytarabine(Ara-C):在體內會受Deoxycytidine kinase轉變成araCTP→抑制DNA合成
會受到Cytodone deaminase代謝→Deoxycytidine kinase/Cytodone deaminase比值可計算濃度及毒性
AML(Ara-C+doxorubicin or mitoxantrone)
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