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Anti-Cancer (DNA Replication Inhibitors (DNA precursors/ antimetabolites …
Anti-Cancer
DNA Replication Inhibitors
DNA precursors/
antimetabolites
(S phase)
Folic Acid
Dihydrofolate reductase inhibitor
aminopterin
methotrexate
pemetrexed
pralatrexate
Thymidylate synthase inhibitor
raltitrexed
pemetrexed
Purine
Adenosine deaminase inhibitor
pentostatin
Halogenated/ribonucleotide reductase inhibitors
cladribine
clofarabine
fludarabine
nelarabine
Thiopurine
mercaptopurine
tioguanine
Pyrimidine
Thymidylate synthase inhibitor
fluorouracil
capecitabine
doxifluridine
Tegafur (+gimeracil/oteracil)
carmofur
floxuridine
DNA polymerase inhibitor
cytarabine
Ribonucleotide reductase inhibitor
gemcitabine
Hypomethylating agent
azacitidine
decitabine
Deoxyribonucleotide
Ribonucleotide reductase inhibitor
hydroxycarbamide
Topoisomerase inhibitors
(S phase)
I
Camptotheca
camptothecin
cositecan
belotecan
gimatecan
exatecan
irinotecan
lurtotecan
silatecan
topotecan
rubitecan
II
Podophyllum
etoposide
teniposide
II+Intercalation
Anthracyclines
aclarubicin
daunorubicin
doxorubicin
epirubicin
idarubicin
amrubicin
pirarubicin
valrubicin
zorubicin
Anthracenediones
mitoxantrone
pixantrone
Crosslinking of DNA
(CCNS)
Alkylating
Nitrogen mustards
mechlorethamine
cyclophosphamide
trofosfamide
ifosfamide
chlorambucil
melphalan
bendamustine
prednimustine
estramustine phosphate
uramustine
Nitrosoureas
carmustine
lomustine
semustine
fotemustine
nimustine
ranimustine
streptozocin
Alkyl sulfonates
busulfan
mannosulfan
treosulfan
Aziridines
carboquone
thiotepa
triaziquone
triethylenemelamine
Platinum-based
carboplatin
cisplatin
dicycloplatin
nedaplatin
oxaliplatin
satraplatin
Nonclassical
Hydrazines
procarbazine
Triazenes
dacarbazine
temozolomide
altretamine
mitobronitol
pipobroman
Intercalation
streptomyces
actinomycin
bleomycin
mitomycins
plicamycin
Other
Enzyme inhibitors
Farnesyltransferase
tipifarnib
Cyclin-dependent kinase
abemaciclib
alvocidib
palbociclib
ribociclib
seliciclib
Proteasome
bortezomib
carfilzomib
ixazomib
Phosphodiesterase
anagrelide
IMP dehydrogenase
tiazofurin
Lipoxygenase
masoprocol
PARP
niraparib
olaparib
rucaparib
veliparib
HDAC
belinostat
panobinostat
romidepsin
Pi3K
idelalisib
Receptor antagonists
Endothelin
atrasentan
Retinoid X
bexarotene
Sex steroid
testolactone
Other/ungrouped
amsacrine
trabectedin
Retinoids
alitretinoin
tretinoin
arsenic trioxide
Asparagine depleters
asparaginase
pegaspargase
celecoxib
demecolcine
elesclomol
elsamitrucin
etoglucid
lonidamine
lucanthone
mitoguazone
mitotane
oblimersen
omacetaxine mepesuccinate
eribulin
Targeted
Her2/Neu
mab
trastuzumab
trastuzumab/emantine (TDM1)
panitumumab
TKI
lapatinib
EGFR
1st Generation
erlotinib
gefitinib
2nd Generation
Spindle Poisons/Mitotic Inhibitor
Block microtubule assembly
Vinca Alkaloids
vinblastine
vincristine
vinflunine
vinorelbine
vindesine
Block microtubule disassembly
Taxanes
cabazitaxel
docetaxel
larotaxel
ortataxel
paclitaxel
tesetaxel
Epothilones
ixabepilone
Photosenstizers