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Hormone Agonists (Oestrogen + Progesterones (MoA (O): recruit mammary…
Hormone Agonists
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GnRH Analogues
MoA: (initial increase then) paradoxial decrease in gonadotrophin due to receptor downregulation in pituitary
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Nasal spray or injection, continuous non-pulsatile
Various sex-hormone dependent conditions, inc. prostate, pre-menopausal breast cancer, endometriosis.
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Somatostatin analogues
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MoA: tumours express receptors, binding activates decreased proliferation and hormone secretion
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