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Lec 11 - Cancer Chemotherapy (Prostate Cancer (GnRH agonist (Leuprolide…
Lec 11 - Cancer Chemotherapy
Alkylating agents
Nitrogen mustards
Cyclophosphamide (Cytoxan)
Mesna
Nitrosureas
Carmustine
Platinum compounds
Cisplatin
Antimetabolites
Folic Acid Analogs
Methotrexate
Leukovorin
Pyrimidine Analogs
Cytarabine (Cytosine arabinoside, Ara-C)
Purine Analogs
Mercaptopurine (Purinethol)
Topoisomerase Inhibitors
Etoposide (Toposar)
Antitumor antibiotics
Anthracyclines
Conventional
Doxorubicin (Adriamycin)
Zinecard
Liposomal
Doxorubicin (Doxil, Caelyx)
Zinecard
Non-Anthracyclines
Dactinomycin (Actinomycin D)
Mitotic Inhibitors
Vinca alkaloids
Conventional
Vincristine (Oncovin)
Liposomal
Vincristine (Marqibo)
Vinblastine (Velban)
Taxanes
Paclitaxel (Taxol)
Asparaginase (Elspar)
Breast Cancer
Anti-estrogens
Tamoxifen
Aromatase inhibitors
Anastrozole
Anti-HER2 Antibodies
Trastuzumab (Herceptin)
Kinase Inhibitor
Lapatinib (Tykerb)
Prostate Cancer
GnRH agonist
Leuprolide (Eligard)
GnRH antagonist
Degarelix (Firmagon)
Androgen receptor blocker
Flutamide
CYP17 Inhibitor
Abiraterone (Zytiga)
Angiogenesis Inhibitor
Bevacizumab (Avastin)